A one pot three-step process for the synthesis of an array of arylated benzimidazoribosyl nucleosides

Jolanta Haluszczak, Simon J. F. Macdonald, Marie E. Migaud

Research output: Contribution to journalArticle

4 Citations (Scopus)

Abstract

A three-step one pot reaction/purification protocol was developed to facilitate rapid access to benzimidazole-based nucleosides, for which benzoylated benzimidazoribosyl nucleosides incorporating boronic esters were key reaction intermediates.

Original languageEnglish
Pages (from-to)2821-2831
Number of pages11
JournalOrganic and Biomolecular Chemistry
Volume9
Issue number8
DOIs
Publication statusPublished - 21 Apr 2011

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nucleosides
Nucleosides
Reaction intermediates
reaction intermediates
synthesis
purification
Purification
esters
Esters
benzimidazole

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Haluszczak, Jolanta ; Macdonald, Simon J. F. ; Migaud, Marie E. / A one pot three-step process for the synthesis of an array of arylated benzimidazoribosyl nucleosides. In: Organic and Biomolecular Chemistry. 2011 ; Vol. 9, No. 8. pp. 2821-2831.
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A one pot three-step process for the synthesis of an array of arylated benzimidazoribosyl nucleosides. / Haluszczak, Jolanta; Macdonald, Simon J. F.; Migaud, Marie E.

In: Organic and Biomolecular Chemistry, Vol. 9, No. 8, 21.04.2011, p. 2821-2831.

Research output: Contribution to journalArticle

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